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E-mail: yamaryu@rs.kagu.tus.ac.jp
2004
@@@ĺwňwn¤ČŞqňwęUmŰöCš@ňwm
2004~2007
@@@Scripps ¤@m¤ő (M. Reza Ghadiri)
i2005 ă´LOś˝Čwŕc@COŻwT[`tF[Vbvj@
2007
@@@ČĺwwćęťwČ@ł@iÄĄTę@yłöj
RYU YAMASAKI
Ph. D.
Assistant Professor
Organic Chemistry
(Peptide, Medicinal, stereo chemistry)
E-mail: yamaryu@rs.kagu.tus.ac.jp
2004
@@@Ph. D. (Pharmaceutical Science), The University of TOKYO, Japan
2004~2007
@@@Post-doctoral Fellow, The Scripps Research Institute (Prof. M. Reza Ghadiri)
i2005 The Uehara Memorial Foundation, Research Fellowshipj@
2007
@@@Assistant Professor, Tokyo University of Science, Japan (Ass. Prof. Shinichi, Saito)
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1, Novel small molecule nonpeptide aminopeptidase N inhibitors with a
cyclic imide skeleton
Rumiko Shimazawa,
Hisae Takayama, Yasuuki Fujimoto, Masato Komoda, Kousuke Dodo, Ryu Yamasaki,
Ryuichi Shirai, Yukiko Koiso, Keizo Miyata, Fuminori, Kato, Masanari Kato,
Hiroyuki Miyachi, Yuichi Hashimoto; J.
Enzyme Inhibition, 1999, 14, 259-275
2,
Novel inhibitors of
alpha-glucosidase with tetrachlorophthalmide skeleton
Sonei Sou, Satoshi
Mayumi, Hiroyasu Takahashi, Ryu Yamasaki, Shizuo Kadoya, Mikiko Sodeoka, Yuichi
Hashimoto; Bioorganic & Medicinal
Chemistry Lett., 2000, 10(10), 1081-1086
3,
Srtucture of N,Nf-bis(1,2-dicarba-closo-dodecaboran-1-yl)-phenylureas:
building blocks for carborane-containing macromolecules
Chalermkiat Songkram,
Aya Tanatani, Ryu Yamasaki, Kentaro Yamaguchi, Hiroyuki Kagechika, Yasuyuki
Endo; Tetrahedron Lett., 2000, 41(36), 7065-7070
4,
a-Glucosidase
Inhibitors with a Phthalimide Skeleton: Structure-Activity Relationship Study
Hiroyasu Takahashi,
Sonei Sou, Ryu Yamasaki, Mikiko Sodeoka, Yuichi Hashimoto; Chem. Pharm. Bull., 2000,
48(10), 1494-1499
5,
a-Glucosidase
Inhibitors with a 4,5,6,7-Tetrachlorophtalimide Skelton Pendanted with a
Cycloalkyl or Dicarba-closo-dodecaborane Group
Sonei Sou, Hiroyasu
Takahashi, Ryu Yamasaki, Hiroyuki Kagechika, Yasuyuki Endo, Yuichi Hashimoto; Chem. Pharm. Bull., 2001, 49(6), 791-793
6,
Molecular construction based on
icosahedral carboranes and aromatic urea groups. A new types of carboracycle
Chalermkiat
Songkram, Ryu Yamasaki, Aya Tanatani, Kojiro Takaishi, Kentaro Yamaguchi, Hiroyuki Kagechika,
Yasuyuki Endo; Tetrahedron Lett., 2001, 42(34), 5913-5916
7,
Molecular construction based on
icosahedral carboranes and aromatic N,N'-dimethylurea groups. Aromatic layered
molecules and a transition metal complex
Yasuyuki Endo, Chalermkiat Songkram, Ryu Yamasaki, Aya Tanatani, Hiroyuki Kagechika, Kojiro Takaishi, Kentaro Yamaguchi; Journal of Organometallic Chem., 2002, 657, 48-58
8,
Amide Conformational Switching Induced by Protonation of Aromatic
Substituent
Ryu Yamasaki, Aya Tanatani, Isao Azumaya, Shoichi
Saito, Kentaro Yamaguchi,
Hiroyuki Kagechika; Organic Letters, 2003, 5(8), 1265-1267
9, Absolute Helical Arrangement of Sulfonamide
in the Crystal
Isao
Azumaya, Takako Kato, Iwao Okamoto, Ryu Yamasaki, Aya Tanatani,
Kentaro Yamaguchi,
Hiroyuki Kagechika; Organic Letters, 2003, 5(21), 3939-3942
10, Solvent-Dependent Conformational Switching
of N-phenylhydrosamic Acid and Its
Application in Crystal Engineering
Ryu Yamasaki, Aya
Tanatani, Isao Azumaya, Hyuma Masu, Kentaro Yamaguchi, Hiroyuki Kagechika; Cryst. Growth. Des., 2006,
6(9), 2007-2010.